Activators & Inhibitors

AMY-101 TFA (Cp40 TFA) is a peptidic inhibitor of the central complement component C3 (KD: 0.5 nM). AMY-101 TFA shows a favorable anti-inflammatory activity in models with COVID-19 severe pneumonia with systemic hyper inflammation.

Ramoplanin is a broad-spectrum lipoglycodepsipeptide antibiotic with activity against gram-positive bacteria. It is existed in the Actinoplanes spp.

Lysipressin Acetate is an analog of vasopressin, a powerful vasopressin used to regulate blood pressure. Endogenous vasopressin in most mammalian species.

(2S,3AS,7aS)-Octahydroindole-2-carboxylic acid is a useful organic compound that has been used in life science related research.

Compound 1769-24-0 is a natural product for research related to life sciences. The catalog number is TPL0186 and the CAS number is 1769-24-0.

4-(Benzo[d]oxazol-2-yl)aniline is a potent antitumor agent that has inhibitory activity against mammary carcinoma cell lines [1].

AP1867-3-(aminoethoxy) is a synthetic ligand for FKBP and can be used in the synthesis of PROTAC FKBP12 F36V degrader.

SLF-amido-C2-COOH is a synthetic ligand for FKBP (SLF), and can be used in the synthesis of PROTACs.

Umbellulone is a natural product isolated from Umbellularia californica, and stimulates the TRPA1 channel in a subset of peptidergic, nociceptive neurons, activating the trigeminovascular system via this mechanism.