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    Results for Activators & Inhibitors ( 75657 )

      • Ref: T62194
        Sizes: 5 mg, 100 mg, 50 mg

        MEIS-IN-3 is a potent inhibitor of MEIS.

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      • Ref: T62195
        Sizes: 5 mg, 100 mg, 50 mg

        Analgesic agent-1 is a potent analgesic that exhibits significant analgesic activity.

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      • Ref: T62196
        Sizes: 5 mg, 100 mg, 50 mg

        CEP-9722 is a prodrug of CEP-8983, a selective, orally active inhibitor of PARP-1 (IC50: 20 nM) and PARP-2 (IC50: 6 nM).CEP-9722 exhibits anticancer activity.

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      • Ref: T62197
        Sizes: 5 mg, 100 mg, 50 mg

        Influenza virus-IN-4 (compound 11e) is a potent inhibitor of influenza virus neuraminidase, acting on H5N1 (IC50: 3.4 μM), H5N2 (IC50: 0.094 μM), H5N6 (IC50: 0.79 μM) and H5N8 (IC50: 0.077 μM). Influenza virus-IN-4 inhibits NA (neuraminidase) and has low cytotoxicity (CC50 > 200 μM). influenza virus-IN-4 is not significantly toxic to mice at 1500 mg/kg.

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      • Ref: T62198
        Sizes: 5 mg, 100 mg, 50 mg

        AR524 is a transgenic inhibitor with higher inhibitory activity than the known transgenic inhibitor kifunensine. AR524 inhibits the formation of human malignant cell spheroids at low concentrations (10 μM).

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      • Ref: T62199
        Sizes: 5 mg, 100 mg, 50 mg

        Talnetant (SB 223412) hydrochloride is a selective NK3 receptor antagonist that acts in hNK-3-CHO cells (Ki: 1.4 nM). Talnetant hydrochloride is 100 times more selective for the hNK-3 receptor than the hNK-2 receptor and has no affinity for hNK-1 at a concentration of 100 μM.

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      • Ref: T62200
        Sizes: 100 mg, 50 mg

        Bunamidine hydrochloride is a veterinary anthelmintic that acts against Echinococcus granulosus and Tapeworm.

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      • Ref: T62201
        Sizes: 5 mg, 100 mg, 50 mg

        TRPC6-IN-2 is a TRPC protein inhibitor, specifically inhibiting TRPC6 protein.

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      • Ref: T62202
        Sizes: 5 mg, 100 mg, 50 mg

        mGluR2 modulator 1 (compound 95) is a potent, blood-brain-barrier permeable modulator of mGluR2 (metabotropic glutamate receptor-2) positive transmutation (EC50: 0.03 μM). mGluR2 modulator 1 can be used in the study of psychiatric disorders.

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